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U 89843A

CAS No. 157013-32-6

U 89843A( —— )

Catalog No. M27731 CAS No. 157013-32-6

U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    U 89843A
  • Note
    Research use only, not for human use.
  • Brief Description
    U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.
  • Description
    U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.(In Vitro):In the alpha 1 beta 2 gamma 2 subtype of GABAA receptors expressed in human embryonic kidney cells, U 89843A dose-dependently enhanced 5 microM GABA-induced Cl- currents with a maximal enhancement of 362 +/- 91%, a half-maximal concentration of 2 +/- 0.4 microM and a slope factor of 1.1 +/- 0.4. U 89843A also inhibited [35S]t-butylbicyclophosphorothionate binding in rat cerebrocortical membranes with a similar half-maximal inhibitory concentration.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    acetylcholinesterase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    157013-32-6
  • Formula Weight
    321.85
  • Molecular Formula
    C16H24ClN5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.Cc1cc2c(nc(nc2n1C)N1CCCC1)N1CCCC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Dafforn A, et al. Acetylcholinesterase inhibition by the ketone transition state analog phenoxyacetone and 1-halo-3-phenoxy-2-propanones. Biochem Biophys Res Commun. 1982 Jan 29;104(2):597-602.
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