Cart
sales@molnova.com
Home - Products - Others - Other Targets - U 89843A

U 89843A

CAS No. 157013-32-6

U 89843A ( —— )

Catalog No. M27731 CAS No. 157013-32-6

U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 873 Get Quote
50MG 1782 Get Quote
100MG 2250 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    U 89843A
  • Note
    Research use only, not for human use.
  • Brief Description
    U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.
  • Description
    U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.(In Vitro):In the alpha 1 beta 2 gamma 2 subtype of GABAA receptors expressed in human embryonic kidney cells, U 89843A dose-dependently enhanced 5 microM GABA-induced Cl- currents with a maximal enhancement of 362 +/- 91%, a half-maximal concentration of 2 +/- 0.4 microM and a slope factor of 1.1 +/- 0.4. U 89843A also inhibited [35S]t-butylbicyclophosphorothionate binding in rat cerebrocortical membranes with a similar half-maximal inhibitory concentration.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    acetylcholinesterase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    157013-32-6
  • Formula Weight
    321.9
  • Molecular Formula
    C16H24ClN5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.Cc1cc2c(nc(nc2n1C)N1CCCC1)N1CCCC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Dafforn A, et al. Acetylcholinesterase inhibition by the ketone transition state analog phenoxyacetone and 1-halo-3-phenoxy-2-propanones. Biochem Biophys Res Commun. 1982 Jan 29;104(2):597-602.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Diacetazotol

    Diacetazotol has activity against dioxin-induced ethoxyisochromamide-O-deethylase (EROD,IC50 = 75±4 nM).

  • N-Succinimidyl 4-(N-...

    N-Succinimidyl 4-(N-maleimidomethyl)cycl(SMCC) also known as succinimidyl-4-[N-maleimidomethyl]cyclohexane-1-carboxylate is a heterobifunctional protein crosslinker.

  • Antennapedia Peptide

    Antennapedia Peptide is a 16 amino acid peptide corresponding to the region within the Drosophila Antennapedia DNA binding domain that is mapped to be responsible for cellular internalization.

Sign In Join Free